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Collaborations and top research areas from the last five years
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RGN6024 Is a Brain-Penetrant, Small-Molecule Tubulin Destabilizer for the Treatment of Glioblastoma
Patrón, L. A., Yeoman, H., Ramos, J., Risinger, A. L., Gokhale, V. & Suzuki, T. C., Aug 1 2025, In: Molecular Cancer Therapeutics. 24, 8, p. 1129-1144 16 p.Research output: Contribution to journal › Article › peer-review
1 Link opens in a new tab Scopus citations -
Role of Human DNA Ligases in Mediating Pharmacological Activities of Flavonoids
Sun, D. & Gokhale, V., Feb 2025, In: International journal of molecular sciences. 26, 4, 1456.Research output: Contribution to journal › Article › peer-review
Open Access1 Link opens in a new tab Scopus citations -
Discovery and Functional Characterization of a Potent, Selective, and Metabolically Stable PROTAC of the Protein Kinases DYRK1A and DYRK1B
Wilms, G., Schofield, K., Maddern, S., Foley, C., Shaw, Y., Smith, B., Basantes, L. E., Schwandt, K., Babendreyer, A., Chavez, T., McKee, N., Gokhale, V., Kallabis, S., Meissner, F., Rokey, S. N., Dunckley, T., Montfort, W. R., Becker, W. & Hulme, C., Oct 10 2024, In: Journal of Medicinal Chemistry. 67, 19, p. 17259-17289 31 p.Research output: Contribution to journal › Article › peer-review
8 Link opens in a new tab Scopus citations -
Novel Brain-Penetrant, Small-Molecule Tubulin Destabilizers for the Treatment of Glioblastoma
Patrón, L. A., Yeoman, H., Wilson, S., Tang, N., Berens, M. E., Gokhale, V. & Suzuki, T. C., Feb 2024, In: Biomedicines. 12, 2, 406.Research output: Contribution to journal › Article › peer-review
Open Access3 Link opens in a new tab Scopus citations -
Quindoline-derivatives display potent G-quadruplex-mediated antiviral activity against herpes simplex virus 1
Frasson, I., Soldà, P., Nadai, M., Tassinari, M., Scalabrin, M., Gokhale, V., Hurley, L. H. & Richter, S. N., Dec 2022, In: Antiviral Research. 208, 105432.Research output: Contribution to journal › Article › peer-review
Open Access12 Link opens in a new tab Scopus citations
Datasets
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In vitro activity of a G-quadruplex-stabilizing small molecule that synergizes with Navitoclax to induce cytotoxicity in acute myeloid leukemia cells
Montoya, J. J. (Creator), Turnidge, M. A. (Creator), Wai, D. H. (Creator), Patel, A. R. (Contributor), Lee, D. W. (Creator), Gokhale, V. (Creator), Hurley, L. H. (Creator), Arceci, R. J. (Creator), Wetmore, C. (Creator) & Azorsa, D. O. (Creator), figshare, 2019
DOI: 10.6084/m9.figshare.c.4799331.v1, https://springernature.figshare.com/collections/In_vitro_activity_of_a_G-quadruplex-stabilizing_small_molecule_that_synergizes_with_Navitoclax_to_induce_cytotoxicity_in_acute_myeloid_leukemia_cells/4799331/1
Dataset
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CCDC 709587: Experimental Crystal Structure Determination
Vardanyan, R. (Creator), Vijay, G. (Creator), Nichol, G. S. (Creator), Liu, L. (Creator), Kumarasinghe, I. (Creator), Davis, P. (Creator), Vanderah, T. (Creator), Porreca, F. (Creator), Lai, J. (Creator) & Hruby, V. J. (Creator), Cambridge Crystallographic Data Centre, 2010
DOI: 10.5517/ccrtcxt, http://www.ccdc.cam.ac.uk/services/structure_request?id=doi:10.5517/ccrtcxt&sid=DataCite
Dataset
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In vitro activity of a G-quadruplex-stabilizing small molecule that synergizes with Navitoclax to induce cytotoxicity in acute myeloid leukemia cells
Montoya, J. J. (Creator), Turnidge, M. A. (Creator), Wai, D. H. (Creator), Patel, A. R. (Contributor), Lee, D. W. (Creator), Gokhale, V. (Creator), Hurley, L. H. (Creator), Arceci, R. J. (Creator), Wetmore, C. (Creator) & Azorsa, D. O. (Creator), figshare, 2019
DOI: 10.6084/m9.figshare.c.4799331, https://springernature.figshare.com/collections/In_vitro_activity_of_a_G-quadruplex-stabilizing_small_molecule_that_synergizes_with_Navitoclax_to_induce_cytotoxicity_in_acute_myeloid_leukemia_cells/4799331
Dataset
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CCDC 843705: Experimental Crystal Structure Determination
Raghunand, N. (Creator), Guntle, G. P. (Creator), Gokhale, V. (Creator), Nichol, G. S. (Creator), Mash, E. A. (Creator) & Jagadish, B. (Creator), Cambridge Crystallographic Data Centre, 2011
DOI: 10.5517/ccx9y9f, http://www.ccdc.cam.ac.uk/services/structure_request?id=doi:10.5517/ccx9y9f&sid=DataCite
Dataset
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Crystal structure of the NM23-H2 transcription factor complex with dinucleotide d(AG)
Dexheimer, T. S. (Contributor), Carey, S. S. (Contributor), Zuohe, S. (Contributor), Gokhale, V. M. (Contributor), Hu, X. (Contributor), Murata, L. B. (Contributor), Maes, E. M. (Contributor), Weichsel, A. (Contributor), Sun, D. (Contributor), Meuillet, E. J. (Contributor), Montfort, W. R. (Contributor), Hurley, L. H. (Contributor), Moréra, S. (Contributor), Lacombe, M.-L. (Contributor), Yingwu, X. (Contributor) & Joël Janin, G. L. A. (Contributor), Protein Data Bank (PDB), Sep 23 2008
DOI: 10.2210/pdb3BBB/pdb, https://www.wwpdb.org/pdb?id=pdb_00003bbb
Dataset